PROTAC ERRα ligand 1

CAS No. 1264754-13-3

PROTAC ERRα ligand 1 ( —— )

Catalog No. M23437 CAS No. 1264754-13-3

PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).

Purity : >98% (HPLC)

COA Datasheet HNMR HPLC MSDS Handing Instructions
Size Price / USD Stock Quantity
2MG 57 In Stock
5MG 87 In Stock
10MG 132 In Stock
25MG 237 In Stock
50MG 385 In Stock
100MG 575 In Stock
500MG 1233 In Stock
1G Get Quote In Stock

Biological Information

  • Product Name
    PROTAC ERRα ligand 1
  • Note
    Research use only, not for human use.
  • Brief Description
    PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
  • Description
    PROTAC ERRα ligand 1 is an α (ERRα) antagonist of estrogen-related receptor (IC50s of 0.04 and 2.8 μM for ERRα and ERRγ, respectively).
  • Synonyms
    ——
  • Pathway
    Endocrinology/Hormones
  • Target
    Estrogen Receptor/ERR
  • Recptor
    ERRα;ERRγ
  • Research Area
    ——
  • Indication
    ——

Chemical Information

  • CAS Number
    1264754-13-3
  • Formula Weight
    420.4
  • Molecular Formula
    C19H11F3N2O4S
  • Purity
    >98% (HPLC)
  • Solubility
    DMSO : 120 mg/mL (285.47 mM; Need ultrasonic)
  • SMILES
    N#CC1=CC=C(OC2=CC=C(/C=C(SC(N3)=O)/C3=O)C=C2OC)C(C(F)(F)F)=C1
  • Chemical Name
    ——

Shipping & Storage Information

  • Storage
    (-20℃)
  • Shipping
    With Ice Pack
  • Stability
    ≥ 2 years

Reference

1.Patch RJ, et al. Identification of diaryl ether-based ligands for estrogen-related receptor α as potential antidiabetic agents. J Med Chem. 2011 Feb 10;54(3):788-808.
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